Epics Therapeutics (former Euroscreen)のEuroscreenFASTでは、Aequorin (カルシウム)、cAMP、GTPγS、IPOne等の様々なアッセイ方法により、GPCR functional Assayが可能です。アゴニスト及びアンタゴニスト活性の測定の他、PAMやNAMの測定も実施しております。様々な種もラインナップされておりますので、種差の検証にも有用です。また、Radioligand bindingアッセイも提供しておりますので、Functional assayと組み合わせての利用も可能です。

FAMILYRECEPTORSPECIESAequorincAMPIPOneGTPgSRadioligand bindingERK1/2Internalisation
AdenosineA1HSFAST-001AFAST-001CFAST-001GFAST-001B
MMFAST-031CFAST-031GFAST-031B
CFFAST-0165CFAST-0165B
RNFAST-0162CFAST-0162B
A2AHSFAST-002AFAST-002CFAST-002GFAST-002B
MMFAST-032CFAST-032B
RNFAST-0163CFAST-0163B
CFFAST-0166CFAST-0166C
A2BHSFAST-003AFAST-003CFAST-003B
MMFAST-033CFAST-033B
RNFAST-0164C
CFFAST-0167C
A3HSFAST-004AFAST-004CFAST-004GFAST-004B
MMFAST-034CFAST-034GFAST-034B
RNFAST-012CFAST-012GFAST-012B
CFFAST-0168C
Adrenergica1AHSFAST-005AFAST-005CFAST-005IFAST-005B
a1BHSFAST-008AFAST-008IFAST-008B
a1DHSFAST-009AFAST-009IFAST-009B
a2AHSFAST-006AFAST-006CFAST-006GFAST-006B
a2BHSFAST-007AFAST-007GFAST-007B
CFFAST-013AFAST-013GFAST-013B
a2CHSES-032AES-032CES-032GES-032B
b1HSES-033AES-033CES-033B
b2HSES-034CES-034B
b3HSES-035AES-035CES-035B
AnaphylotaxinC3aHSFAST-010AFAST-010CFAST-010GFAST-010B
C5aHSFAST-011CFAST-011G
C5a2 (C5AR2/GPR77)HSFAST-0960B
AngiotensinAT1HSFAST-015AFAST-015IFAST-015B
CFFAST-037B
AT2HSFAST-016B
MMFAST-017B
CFFAST-038B
ApelinAPJHSFAST-020AFAST-020CFAST-020GFAST-020B
Bile AcidGPBA (TGR5/GPR131)HSFAST-0965C
CFFAST-0966C
MMFAST-0967C
RNFAST-0968C
BombesinBB1HSFAST-022AFAST-022B
BB2HSFAST-023AFAST-023B
BB3HSFAST-021AFAST-021B
MMFAST-018***
RNFAST-019***
BradykininB1HSFAST-027AFAST-027IFAST-027B
RNFAST-0207A
B2HSFAST-028AFAST-028B
CalcitoninCGRP (CRLR/RAMP1)HSFAST-025AFAST-025CFAST-025B
MMFAST-054C
RNFAST-055C
AM1 (CRLR/RAMP2)HSFAST-026C
AM2 (CRLR/RAMP3)HSFAST-024AFAST-024CFAST-024B
AMY1 (CTR/RAMP1)HSFAST-035C
AMY2 (CTR/RAMP2)HSFAST-036C
AMY3 (CTR/RAMP3)HSFAST-029CFAST-029B
CTRHSFAST-030C
CalciumCaSHSFAST-0680AFAST-0680I
CannabinoidCB1HSFAST-040CFAST-040GFAST-040BFAST-040E
RNFAST-044CFAST-044GFAST-044B
MFFAST-042C
OCFAST-046C
CB2HSFAST-041CFAST-041GFAST-041B
RNFAST-045CFAST-045GFAST-045B
ChemerinCCRL2HSFAST-0948B
CMKLR1 (ChemR23)HSFAST-050AFAST-050CFAST-050GFAST-050BFAST-050E
CMKLR1 (ChemR23)RNFAST-053A
CMKLR1 (DEZ)MMFAST-051AFAST-051B
GPR1HSFAST-052B
ChemokineCCR1HSFAST-058AFAST-058CFAST-058GFAST-058B
MMFAST-059C
CCR2bHSFAST-060AFAST-060CFAST-060GFAST-060B
MMFAST-0600AFAST-0600CFAST-0600B
RNFAST-0616AFAST-0616CFAST-0616B
RHFAST-0710AFAST-0710B
CCR3HSFAST-061AFAST-061GFAST-061B
MMFAST-0601A
CCR4HSFAST-069AFAST-069CFAST-069GFAST-069B
MMFAST-0602A
CCR5*HSFAST-062AFAST-062CFAST-062GFAST-062BFAST-062E
MMFAST-0603AFAST-0603CFAST-0603B
RNFAST-0617AFAST-0617CFAST-0617B
CFFAST-0712A
RHFAST-0711AFAST-0711CFAST-0711B
OCFAST-0713A
CCR6HSFAST-063AFAST-063CFAST-063GFAST-063B
MMFAST-0604AFAST-0604C
CCR7HSFAST-064AFAST-064CFAST-064GFAST-064BFAST-064E
MMFAST-0605A
CCR8HSFAST-065AFAST-065CFAST-065GFAST-065B
MMFAST-0606AFAST-0606C
CCR9aHSFAST-066A
MMFAST-0607A
CCR10HSFAST-067AFAST-067CFAST-067G
MMFAST-0608A
CXCR1HSFAST-071AFAST-071CFAST-071GFAST-071B
MMFAST-0609A
CXCR2HSFAST-075AFAST-075CFAST-075GFAST-075B
MMFAST-0610A
CXCR3aHSFAST-076AFAST-076GFAST-076B
MMFAST-0611A
CXCR3bHSFAST-0761A
CXCR4HSFAST-077AFAST-077CFAST-077GFAST-077B
MMFAST-0612A
RNFAST-0619A
CXCR5HSFAST-078AFAST-078G
MMFAST-0613A
CXCR6HSFAST-080AFAST-080CFAST-080G
MMFAST-0614A
CXCR7HSFAST-081B
CX3CR1HSFAST-070AFAST-070CFAST-070GFAST-070BFAST-070E
MMFAST-0615AFAST-0615G
RNFAST-0618A
XCR1HSFAST-085AFAST-085CFAST-085G
CholecystokininCCK1HSFAST-090AFAST-090CFAST-090IFAST-090B
CCK2HSFAST-091AFAST-091IFAST-091B
Corticotropin-releasing factorCRF1HSFAST-095AFAST-095CFAST-095GFAST-095B
CRF2aHSFAST-097C
RNFAST-098C
CFFAST-094C
CRF2bHSFAST-096CFAST-096B
DopamineD1HSFAST-0100CFAST-0100B
RNFAST-0126C
D2LHSFAST-0101AFAST-0101CFAST-0101GFAST-0101B
D2SHSFAST-0102AFAST-0102CFAST-0102GFAST-0102B
MMFAST-0132C
RNFAST-0127C
D3HSES-173GES-173B
D4.4HSFAST-099CFAST-099GFAST-099B
RNFAST-0103GFAST-0103B
D5HSFAST-0104C
RNFAST-0129C
EndothelinETAHSFAST-0105AFAST-0105B
RNFAST-0107A
ETBHSFAST-0106AFAST-0106B
RNFAST-0108A
FormylpeptideFPR1 (fMLP)HSFAST-0342AFAST-0342C
MMFAST-0345C
OCFAST-0339C
FPR2 (FPRL1)HSFAST-0340AFAST-0340CFAST-0340GFAST-0340B
MMFAST-0343C
RNFAST-0344C
CFFAST-0347C
OCFAST-0348C
MFFAST-0349C
FPR3 (FPRL2)HSFAST-0341AFAST-0341C
Free fatty acidFFA1 (GPR40)HSFAST-0110AFAST-0110I
MMFAST-0109A
FFA3 (GPR41)HSFAST-0111AFAST-0111CFAST-0111G
MMFAST-0118C
FFA2 (GPR43)*HSFAST-0112AFAST-0112CFAST-0112IFAST-0112GFAST-0112E
MMFAST-0116AFAST-0116CFAST-0116IFAST-0116G
RNFAST-0117AFAST-0117CFAST-0117IFAST-0117G
RHFAST-0124AFAST-0124C
CFFAST-0123AFAST-0123C
SSFAST-0125G
GPR35HSFAST-0915AFAST-0915CFAST-0915GFAST-0915E
MMFAST-0991AFAST-0991C
RNFAST-0992AFAST-0992C
GPR84HSFAST-0935AFAST-0935CFAST-0935GFAST-0935EFAST-0935T
MMFAST-0993AFAST-0993C
RNFAST-0994AFAST-0994C
FFA4 (GPR120)HSFAST-0113AFAST-0113IFAST-0113E
MMFAST-0114A
RNFAST-0115A
GABAGABA B1a/B2HSFAST-0120AFAST-0120CFAST-0120GFAST-0120B
GABA B1b/B2HSFAST-0122C
GABA (non-selective)RNFAST-0121B
GalaninGAL1HSFAST-0130AFAST-0130CFAST-0130GFAST-0130B
GAL2HSFAST-0131AFAST-0131IFAST-0131GFAST-0131B
GhrelinGHS-RHSFAST-0135AFAST-0135IFAST-0135B
GlucagonGlucagonHSFAST-0138AFAST-0138CFAST-0138B
MMFAST-0137C
GIPHSFAST-0139AFAST-0139CFAST-0139BFAST-0139T
GLP-1HSFAST-0145AFAST-0145CFAST-0145BFAST-0145T
MMFAST-0147CFAST-0147BFAST-0147T
GLP-2HSFAST-0146C
GHRHRHSFAST-0160C
SecretinHSFAST-0161AFAST-0161C
Glutamate (metabotropic)mGlu1HSFAST-0152AFAST-0152CFAST-0152B
mGlu2HSFAST-0153C
mGlu3HSFAST-0155A
mGlu4HSFAST-0150CFAST-0150G
mGlu5HSFAST-0151AFAST-0151IFAST-0151B
RNFAST-0158B
mGlu6HSFAST-0157G
mGlu7HSFAST-0154C
mGlu8HSFAST-0156G
Glycoprotein hormoneFSHHSFAST-0580C
LHHSFAST-0581C
TSHHSFAST-0582C
MMFAST-0584C
RNFAST-0585C
GnRHGnRHR1HSFAST-0583AFAST-0583B
GPR/OrphanGPR3HSFAST-0700C***
MMFAST-0703C***
RNFAST-0704C***
GPR6HSFAST-0701C***
GPR12HSFAST-0702C***
GPR17HSFAST-0903AFAST-0903CFAST-0903IFAST-0903GFAST-0903T
GPR17longHSFAST-0996AFAST-0996CFAST-0996IFAST-0996G
GPR17MMFAST-0997AFAST-0997CFAST-0997IFAST-0997G
GPR17RNFAST-0998AFAST-0998CFAST-0998IFAST-0998G
GPR18HSFAST-0904***
GPR19 (GPR-NGA)HSFAST-0905***
GPR20HSFAST-0906***
GPR21HSFAST-0907C***
GPR22HSFAST-0908***
GPR23 (LPAR4)HSFAST-0640***
GPR25HSFAST-0909***
GPR26HSFAST-0970C***
GPR27 (SREB1)HSFAST-0910***
GPR30 (GPER)HSFAST-0911A
MMFAST-0886A
RNFAST-0887A
GPR31HSFAST-0912***
GPR32HSFAST-0913***
GPR37HSFAST-0916***
GPR37L1HSFAST-0917***
GPR39HSFAST-0918AFAST-0918C
MMFAST-0932AFAST-0932C
RNFAST-0999C
GPR45HSFAST-0919***
GPR50HSFAST-0920***
GPR52HSFAST-0921C
MMFAST-0891C
RNFAST-0961C
GPR61HSFAST-0924C***
GPR63HSFAST-0925***
GPR75HSFAST-0930***
GPR78HSFAST-0931C***
GPR82HSFAST-0933***
GPR83 (GPR72)HSFAST-0934AFAST-0934I
MMFAST-0945AFAST-0945I
GPR87 (HG03)HSFAST-0937***
GPR88*HSFAST-0938AFAST-0938C
MMFAST-0963C
RNFAST-0964C
GPR101HSFAST-0941C***
MMFAST-0953C***
RNFAST-0954C***
GPR132 (G2A)HSFAST-0967***
GPR139HSFAST-0980A
GPR141HSFAST-0981***
GPR142HSFAST-0969I
MMFAST-0898I
RNFAST-0899I
GPR142 long isoformMMFAST-0896I
RNFAST-0897I
GPR146HSFAST-0976***
GPR148HSFAST-0982***
GPR149HSFAST-0983***
GPR150HSFAST-0984***
GPR151HSFAST-0985***
GPR152HSFAST-0942***
GPR153HSFAST-0978***
GPR161 (RE2)HSFAST-0962C***
GPR162 (A-2)HSFAST-0943***
GPR173 (SREB3)HSFAST-0977***
GPR174 (DA6)HSFAST-0944***
GPR171 (H963)HSFAST-0946***
GPR176 (HB954)HSFAST-0947***
GPR182 (HSGPCP)HSFAST-0949***
GPRC5A (RAIG1)HSFAST-0955***
GPRC5B (RAIG2)HSFAST-0956***
GPRC5C (RAIG3)HSFAST-0957***
GPRC5D (RAIG4)HSFAST-0958***
LGR4HSFAST-0972***
LGR5HSFAST-0973***
LGR6HSFAST-0974***
P2Y5HSFAST-0950***
P2Y8HSFAST-0986A
P2Y10HSFAST-0951***
HistamineH1HSFAST-0170AFAST-0170IFAST-0170B
H2HSFAST-0171AFAST-0171CFAST-0171B
H3*HSFAST-0172AFAST-0172CFAST-0172GFAST-0172B
RNFAST-0174GFAST-0174B
CFFAST-0175G
H4HSFAST-0173AFAST-0173GFAST-0173B
MMFAST-0169G
Hydroxycarboxylic acidGPR109a (HM74a/HCA2)HSFAST-0350AFAST-0350CFAST-0350GFAST-0350B
GPR109b (HM74/HCA3)HSFAST-0351AFAST-0351CFAST-0351GFAST-0351E
GPR81 (HCA1)HSFAST-0352AFAST-0352CFAST-0352G
MMFAST-0353C
RNFAST-0354C
KiSS1/KisspeptinGPR54 (KiSS1)HSFAST-0180AFAST-0180B
RNFAST-0181A
LeukotrieneBLT1 (LTB4R)HSFAST-0192AFAST-0192G
BLT2 (LTB4R2)HSFAST-0194A
CysLT1HSFAST-0190AFAST-0190B
CysLT2*HSFAST-0191AFAST-0191IFAST-0191B
OXE (HM74like)HSFAST-0193A
LysophospholipidsLPA3 (EDG7)HSFAST-0632AFAST-0632I
LPA5 (GPR92)HSFAST-0641I
GPR34HSFAST-0914AFAST-0914CFAST-0914G
GPR55HSFAST-0922AFAST-0922T
Mas relatedMrgX1HSFAST-0213A
MrgX2HSFAST-0214A
MASHSFAST-0210A
MRGHSFAST-0211**
MRGD (TGR7)HSFAST-0212AFAST-0212CFAST-0212G
MRGEHSFAST-0216***
MRGF (RTA)HSFAST-0215***
MelaninMCH1HSFAST-0220AFAST-0220CFAST-0220GFAST-0220B
concentratingMMFAST-0660A
hormoneMCH2HSFAST-0221AFAST-0221B
MelanocortinMC1HSFAST-0230CFAST-0230B
RNFAST-0224C
SSFAST-0225C
MC2 (MC2/MRAP)HSFAST-0231AFAST-0231C
RNFAST-0226C
MC3HSFAST-0232CFAST-0232B
MMFAST-0235C
RNFAST-0227C
SSFAST-0228C
MC4HSFAST-0233CFAST-0233IFAST-0233B
RNFAST-0229C
MC5HSFAST-0234CFAST-0234B
MMFAST-0236CFAST-0236B
RNFAST-0237CFAST-0237B
CFFAST-0238CFAST-0238B
MelatoninMT1HSFAST-0240AFAST-0240GFAST-0240B
MT2HSFAST-0241AFAST-0241GFAST-0241B
MotilinMTLHSFAST-0250AFAST-0250IFAST-0250B
MuscarinicM1HSFAST-0260AFAST-0260IFAST-0260GFAST-0260B
RNFAST-0262A
M2HSFAST-0261AFAST-0261CFAST-0261GFAST-0261B
RNFAST-0263A
M3HSES-212AES-212IES-212B
RNFAST-0266A
M4HSES-213AES-213GES-213B
RNFAST-0267A
M5HSFAST-0264AFAST-0264IFAST-0264B
RNFAST-0268A
Non-selectiveRNFAST-0265B
NeurokininNK1HSFAST-0269AFAST-0269B
MMFAST-0621AFAST-0621B
RNFAST-0622AFAST-0622B
RHFAST-0634A
NK2HSFAST-0270AFAST-0270B
MMFAST-0623A
RNFAST-0624A
RHFAST-0635A
Neuromedin UNMU-1R (FM3)HSFAST-0280AFAST-0280IFAST-0280B
MMFAST-0282I
NMU-2R (FM4)HSFAST-0281AFAST-0281IFAST-0281B
MMFAST-0283IFAST-0283B
NeuropeptideNPY1HSFAST-0320AFAST-0320CFAST-0320GFAST-0320B
RNFAST-0318AFAST-0318C
MFFAST-0319AFAST-0319C
NPY2CFFAST-0333B
HSFAST-0321AFAST-0321CFAST-0321B
MMFAST-0332B
RNFAST-0324AFAST-0324CFAST-0324B
SSFAST-0334B
MFFAST-0325AFAST-0325CFAST-0325B
NPY4HSFAST-0323AFAST-0323CFAST-0323B
RNFAST-0326AFAST-0326C
MFFAST-0327AFAST-0327C
NPY5HSFAST-0322AFAST-0322CFAST-0322B
RNFAST-0328A
MFFAST-0329AFAST-0329C
GPR7HSFAST-0290AFAST-0290CFAST-0290GFAST-0290B
MMFAST-0291A
RNFAST-0292A
GPR8HSFAST-0310AFAST-0310CFAST-0310GFAST-0310B
NPFF1HSFAST-0412CFAST-0412GFAST-0412B
NPFF2SHSFAST-0295AFAST-0295GFAST-0295B
NPS (Ile)HSFAST-0301AFAST-0301B
NPS (Asn)HSFAST-0300AFAST-0300IFAST-0300B
QRFP (GPR103)HSFAST-0302A
NeurotensinNTS1HSFAST-0330AFAST-0330CFAST-0330IFAST-0330GFAST-0330B
NTS2HSFAST-0331AFAST-0331IFAST-0331B
NMDAGRIN1HSFAST-0361B
NociceptinORL1HSFAST-0360CFAST-0360GFAST-0360B
RNFAST-0362B
OleoylethanolamideGPR119*HSFAST-0370C
OpioidOP1 (d)HSFAST-0379AFAST-0379CFAST-0379GFAST-0379B
RNFAST-0378C
OP2 (k)HSFAST-0380AFAST-0380CFAST-0380GFAST-0380B
MMFAST-0375C
RNFAST-0376C
OP3 (µ)HSFAST-0381AFAST-0381CFAST-0381GFAST-0381BFAST-0381E
MMFAST-0382CFAST-0382G
RNFAST-0383CFAST-0383GFAST-0383B
OrexinOX1HSFAST-0390AFAST-0390IFAST-0390B
MMFAST-0394A
RNFAST-0392AFAST-0392I
OX2HSFAST-0391AFAST-0391IFAST-0391B
MMFAST-0395A
RNFAST-0393AFAST-0393I
ParathyroidPTH1HSFAST-0140C
hormonePTH2HSFAST-0141C
pH sensingGPR4HSFAST-0901C
MMFAST-0883C
RNFAST-0884C
CFFAST-0885C
GPR65HSFAST-0927CFAST-0927I
MMFAST-0929C
RNFAST-0880C
GPR68 (OGR1)HSFAST-0928CFAST-0928I
MMFAST-0881C
RNFAST-0882C
Platelet-Activating FactorPAFHSFAST-0650AFAST-0650C
ProkineticinPKR1HSFAST-0400AFAST-0400CFAST-0400B
PKR2HSFAST-0401AFAST-0401CFAST-0401IFAST-0401B
Prolactin-releasing peptidePrRP (GPR10)HSFAST-0410A
ProstanoidDP2/CRTH2HSFAST-0420AFAST-0420CFAST-0420GFAST-0420B
DPHSFAST-0430AFAST-0430CFAST-0430B
EP1HSFAST-0432AFAST-0432B
EP2HSFAST-0443CFAST-0443BFAST-0443E
EP3HSFAST-0444AFAST-0444B
EP4HSFAST-0431AFAST-0431CFAST-0431B
FPHSFAST-0433I
IP1HSFAST-0434CFAST-0434I
TPHSFAST-0438AFAST-0438I
Protease-activatedPAR1HSFAST-0439AFAST-0439IFAST-0439G
PAR2HSFAST-0440AFAST-0440IFAST-0440G
PAR3HSFAST-0441A
PAR4HSFAST-0442A
PurinergicP2Y1HSFAST-0452I
P2Y2HSFAST-0453I
P2Y4*HSFAST-0454I
P2Y6HSFAST-0455AFAST-0455I
P2Y6MMFAST-0459I
P2Y11*HSFAST-0456A
P2Y12HSFAST-0458A
P2Y14HSFAST-0959G
RelaxinRXFP1HSFAST-0469C
MMFAST-0464C
RNFAST-0465C
CFFAST-0466C
OCFAST-0467C
SSFAST-0468C
RXFP3 (GPCR135)HSFAST-0470AFAST-0470CFAST-0470G
RXFP4 (GPCR142)HSFAST-0471AFAST-0471CFAST-0471G
MMFAST-0473G
Serotonin5-HT1AHSFAST-0500AFAST-0500CFAST-0500GFAST-0500B
MMFAST-0475GFAST-0475B
RNFAST-0515GFAST-0515B
CFFAST-0476GFAST-0476B
OCFAST-0477GFAST-0477B
5-HT1BHSFAST-0501CFAST-0501GFAST-0501B
MMFAST-0478GFAST-0478B
RNFAST-0516CFAST-0516GFAST-0516B
CFFAST-0479GFAST-0479B
MFFAST-0474CFAST-0474GFAST-0474B
OCFAST-0480B
5-HT1DHSFAST-0502AFAST-0502GFAST-0502B
MMFAST-0481AFAST-0481B
RNFAST-0482AFAST-0482B
CFFAST-0483B
OCFAST-0484B
5-HT1EHSFAST-0503CFAST-0503GFAST-0503B
CFFAST-0485B
OCFAST-0486B
5-HT1FHSFAST-0504CFAST-0504GFAST-0504B
MMFAST-0487B
RNFAST-0488B
CFFAST-0489GFAST-0489B
OCFAST-0490GFAST-0490B
5-HT2AHSFAST-0505AFAST-0505IFAST-0505B
MMFAST-0491IFAST-0491B
RNFAST-0517AFAST-0517IFAST-0517B
CFFAST-0492IFAST-0492B
OCFAST-0493IFAST-0493B
5-HT2BHSFAST-0506AFAST-0506IFAST-0506B
RNFAST-0518AFAST-0518I
5-HT2C non editedHSFAST-0508AFAST-0508IFAST-0508B
MMFAST-0496I
RNFAST-0519AFAST-0519IFAST-0519B
5-HT2C editedHSFAST-0507AFAST-0507IFAST-0507B
5-HT3HSFAST-0512AFAST-0512B
5-HT4eHSFAST-0513CFAST-0513B
RNFAST-0495C
5-HT5aHSFAST-0510AFAST-0510B
5-HT6HSFAST-0509AFAST-0509CFAST-0509B
MMFAST-0590CFAST-0590B
RNFAST-0494C
5-HT7aHSFAST-0511CFAST-0511B
MMFAST-0498CFAST-0498B
RNFAST-0499CFAST-0499B
Sigmas1HSFAST-0514B
Somatostatinsst1HSFAST-0520GFAST-0520B
sst2HSFAST-0521AFAST-0521CFAST-0521GFAST-0521B
sst3HSFAST-0522AFAST-0522CFAST-0522GFAST-0522B
sst4HSFAST-0523AFAST-0523CFAST-0523GFAST-0523B
RNFAST-0525C
sst5HSFAST-0524AFAST-0524CFAST-0524GFAST-0524B
SphingosineS1P1 (Edg1)HSFAST-0197AFAST-0197CFAST-0197G
MMFAST-0625A
RNFAST-0202AFAST-0202C
FSFAST-0203A
CPFAST-0627A
S1P2 (Edg5)HSFAST-0198A
S1P3 (Edg3)HSFAST-0199A
CPFAST-0628A
S1P4(Edg6)HSFAST-0200AFAST-0200T
S1P5(Edg8)HSFAST-0201AFAST-0201GFAST-0201E
MMFAST-0626A
FSFAST-0204A
CPFAST-0629A
Succinate/Keto glutarateGPR91HSFAST-0450AFAST-0450C
MMFAST-0449AFAST-0449C
RNFAST-0451AFAST-0451C
GPR99HSFAST-0940A
Trace amineTAAR1 (TA1)HSFAST-0987C
MMFAST-0894C
RNFAST-0895C
MFFAST-0893C
TAAR2 (GPR58)HSFAST-0923***
TAAR5 (PNR)HSFAST-0952***
TAAR6 (TA4)HSFAST-0989***
TAAR8 (TA5)HSFAST-0990***
TAAR9 (TA3)HSFAST-0988***
TRHTRH1HSFAST-0530AFAST-0530IFAST-0530B
Tyrosine kinase receptorEGFRHSFAST-1600A
Urotensin IIUT-IIHSFAST-0540AFAST-0540IFAST-0540B
RNFAST-0541A
VasopressinV1aHSFAST-0550AFAST-0550IFAST-0550B
MMFAST-0546A
RNFAST-0555AFAST-0555I
CFFAST-0556AFAST-0556I
OCFAST-0547A
V1bHSFAST-0551AFAST-0551IFAST-0551B
RNFAST-0553IFAST-0553B
V2HSFAST-0552AFAST-0552CFAST-0552IFAST-0552B
RNFAST-0557C
CFFAST-0558C
OT (oxytocin)HSFAST-0554AFAST-0554I
MMFAST-0548A
RNFAST-0559AFAST-0559I
OCFAST-0549A
VIP/PACAPPAC1HSFAST-0560AFAST-0560C
VPAC1HSFAST-0561AFAST-0561CFAST-0561BFAST-0561E
VPAC2HSFAST-0562AFAST-0562C
HS = Homo sapiens ; MM = Mus musculus ; RN = Rattus norvegicus ; CF = Canis familiaris ; CP = Guinea Pig (Cavia porcellus) ; RH = Rhesus monkey (Macaca mulatta) ; OC = Rabbit (Oryctolagus cuniculus) ; MF = Macaca fascicularis ; SS = Pig (Sus scrofa) ; FS = Cat (Felis silvestris catus) ; MA = Syrian hamster (Mesocricetus auratus)
*: Receptors could have limited access due to patent restrictions in certain territories
**: this assay is performed using fluorescent calcium measurement
***: means that the cell line is available for functional assay. It has been validated for mRNA, cell surface expression and constitutive activity but not with a ligand